The safety and scientific validity of this study is the responsibility of the study sponsor and investigators. Listing a study does not mean it has been endorsed by the ANZCTR. Before participating in a study, talk to your health care provider and refer to this information for consumers
Trial details imported from ClinicalTrials.gov

For full trial details, please see the original record at https://clinicaltrials.gov/study/NCT06706076




Registration number
NCT06706076
Ethics application status
Date submitted
19/11/2024
Date registered
26/11/2024
Date last updated
5/09/2025

Titles & IDs
Public title
A Study of BH-30643 in Subjects With Locally Advanced or Metastatic NSCLC Harboring EGFR and/or HER2 Mutations
Scientific title
A Phase 1/2 Open-Label, Multicenter, First-in-Human Study of the Safety, Tolerability, Pharmacokinetics, and Antitumor Activity of BH-30643 in Adult Subjects With Locally Advanced or Metastatic NSCLC Harboring EGFR and/or HER2 Mutations (SOLARA)
Secondary ID [1] 0 0
BH-30643-01
Universal Trial Number (UTN)
Trial acronym
SOLARA
Linked study record

Health condition
Health condition(s) or problem(s) studied:
NSCLC (Advanced Non-small Cell Lung Cancer) 0 0
Condition category
Condition code
Cancer 0 0 0 0
Lung - Non small cell

Intervention/exposure
Study type
Interventional
Description of intervention(s) / exposure
Treatment: Drugs - BH-30643
Treatment: Drugs - BH-30643

Experimental: Phase 1 Dose Escalation and Expansion - * BH-30643 monotherapy for dose escalation
* BH-30643 monotherapy for dose expansion/optimization at doses determined from dose escalation data
* BH-30643 twice daily oral dosing

Experimental: Phase 2 - BH-30643 administered at the RP2D dose determined in Phase 1


Treatment: Drugs: BH-30643
BH-30643 will be provided as either 10 mg or 40 mg capsules. Subjects will take BH-30643 orally depending on their dose level assignment.

Treatment: Drugs: BH-30643
BH-30643 will be provided as either 10 mg or 40 mg capsules. Subjects will take BH-30643 orally depending on their dose level assignment.

Intervention code [1] 0 0
Treatment: Drugs
Comparator / control treatment
Control group

Outcomes
Primary outcome [1] 0 0
Dose-limiting toxicities (DLTs) (Phase 1, Dose Escalation)
Timepoint [1] 0 0
Within the first 21 days of the first dose of BH-30643.
Primary outcome [2] 0 0
Recommended Phase 2 dose (RP2D) (Phase 1, Dose Expansion/Optimization)
Timepoint [2] 0 0
Within 21 days of last participant dosed during Dose Expansion/Optimization.
Primary outcome [3] 0 0
Objective Response Rate (ORR) (Phase 2)
Timepoint [3] 0 0
Approximately 3 years after the first participant dosed.
Secondary outcome [1] 0 0
Safety
Timepoint [1] 0 0
From enrollment through study completion, approximately 48 months.
Secondary outcome [2] 0 0
Area under the plasma concentration-time curve from time zero to time of the last quantifiable concentration (AUClast) of BH-30643 for Single dose (Phase 1).
Timepoint [2] 0 0
Predose and up to 24 hours postdose.
Secondary outcome [3] 0 0
Maximum observed plasma concentration (Cmax) of BH-30643 for Single dose (Phase 1).
Timepoint [3] 0 0
Predose and up to 24 hours postdose.
Secondary outcome [4] 0 0
Time to reach Cmax (Tmax) of BH-30643 for Single dose (Phase 1).
Timepoint [4] 0 0
Predose and up to 24 hours postdose.
Secondary outcome [5] 0 0
Area under the plasma concentration-time curve at steady state (AUCss) of BH-30643 for multiple doses (Phase 1) at steady state.
Timepoint [5] 0 0
Predose and up to 24 hours postdose.
Secondary outcome [6] 0 0
Objective Response Rate (ORR)
Timepoint [6] 0 0
From enrollment until the date of the first documented progression or death from any cause, whichever occurs first, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [7] 0 0
Disease Control Rate (DCR)
Timepoint [7] 0 0
From enrollment until the date of the first documented progression or death from any cause, whichever occurs first, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [8] 0 0
Clinical benefit Rate (CBR)
Timepoint [8] 0 0
From enrollment until the date of the first documented progression or death from any cause, whichever occurs first, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [9] 0 0
Time to Tumor Response (TTR)
Timepoint [9] 0 0
From first dose to the first occurrence of response, assessed up to the date of first documented progression or death from any cause, whichever occurs first (up to approximately 4 years).
Secondary outcome [10] 0 0
Duration of Response (DOR)
Timepoint [10] 0 0
From first occurrence of response until the date of the first documented progression or death from any cause, whichever occurs first, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [11] 0 0
Progression-free Survival (PFS)
Timepoint [11] 0 0
From enrollment until the date of the first documented progression or death from any cause, whichever occurs first, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [12] 0 0
Overall Survival
Timepoint [12] 0 0
From enrollment until the date of death from any cause, assessed up to study ends or patient discontinue from the study, whichever occurs first (up to approximately 4 years).
Secondary outcome [13] 0 0
ERTC-QLC-C30
Timepoint [13] 0 0
From enrollment until the end of treatment, up till patient discontinue from treatment due to any reason (up to approximately 4 years).
Secondary outcome [14] 0 0
NSCLC-SAQ
Timepoint [14] 0 0
From enrollment until the end of treatment, up till patient discontinue from treatment due to any reason (up to approximately 4 years).

Eligibility
Key inclusion criteria
* = 18 years or legal adult.
* Pathologically confirmed diagnosis of locally advanced or metastatic NSCLC with EGFR (classical, atypical, exon20 insertion) or HER2 mutations in the kinase domain of exons 18, 19, 20, or 21. EGFR mutations include activating and acquired EGFR resistance mutations that might form compound mutations.
* Had received standard therapies.
* Has at least 1 measurable target extracranial lesion according to RECIST v1.1.
* Eastern Cooperative Oncology Group Performance Status = 1.
* Has a life expectancy of = 3 months.
* Has adequate hematologic, hepatic, and renal function. *The above are a summary; other Inclusion Criteria details may apply.
Minimum age
18 Years
Maximum age
No limit
Sex
Both males and females
Can healthy volunteers participate?
No
Key exclusion criteria
* History of any concurrent malignancy within the previous 2 years.
* Known other oncogenic driver alterations (eg, moderate or high MET amplification) or histological transformation (eg, to small cell carcinoma, etc.).
* Unresolved toxicities from prior therapies.
* Any significant and uncontrolled medical condition, such as infection.
* History of interstitial lung disease from any cause
* Clinically significant cardiovascular event within 6 months or significant history of major organ.
* Actively receiving investigational therapy(ies) in another clinical study. *The above are a summary; other Exclusion Criteria details may apply.

Study design
Purpose of the study
Treatment
Allocation to intervention
Non-randomised trial
Procedure for enrolling a subject and allocating the treatment (allocation concealment procedures)
Methods used to generate the sequence in which subjects will be randomised (sequence generation)
Masking / blinding
Open (masking not used)
Who is / are masked / blinded?



Intervention assignment
Single group
Other design features
Phase
Phase 1
Type of endpoint/s
Statistical methods / analysis

Recruitment
Recruitment status
Recruiting
Data analysis
Reason for early stopping/withdrawal
Other reasons
Date of first participant enrolment
Anticipated
Actual
Date of last participant enrolment
Anticipated
Actual
Date of last data collection
Anticipated
Actual
Sample size
Target
Accrual to date
Final
Recruitment in Australia
Recruitment state(s)
VIC
Recruitment hospital [1] 0 0
Austin Health - Heidelberg
Recruitment hospital [2] 0 0
Peter MacCallum Cancer Centre - Melbourne
Recruitment postcode(s) [1] 0 0
3084 - Heidelberg
Recruitment postcode(s) [2] 0 0
3000 - Melbourne
Recruitment outside Australia
Country [1] 0 0
United States of America
State/province [1] 0 0
Arizona
Country [2] 0 0
United States of America
State/province [2] 0 0
California
Country [3] 0 0
United States of America
State/province [3] 0 0
Florida
Country [4] 0 0
United States of America
State/province [4] 0 0
Illinois
Country [5] 0 0
United States of America
State/province [5] 0 0
Massachusetts
Country [6] 0 0
United States of America
State/province [6] 0 0
Michigan
Country [7] 0 0
United States of America
State/province [7] 0 0
Minnesota
Country [8] 0 0
United States of America
State/province [8] 0 0
Pennsylvania
Country [9] 0 0
United States of America
State/province [9] 0 0
Tennessee
Country [10] 0 0
United States of America
State/province [10] 0 0
Texas
Country [11] 0 0
United States of America
State/province [11] 0 0
Virginia
Country [12] 0 0
Hong Kong
State/province [12] 0 0
New Territories
Country [13] 0 0
Japan
State/province [13] 0 0
Chiba
Country [14] 0 0
Japan
State/province [14] 0 0
Osaka
Country [15] 0 0
Japan
State/province [15] 0 0
Tokyo
Country [16] 0 0
Singapore
State/province [16] 0 0
Kent Ridge

Funding & Sponsors
Primary sponsor type
Commercial sector/industry
Name
BlossomHill Therapeutics
Address
Country

Ethics approval
Ethics application status

Summary
Brief summary
Trial website
Trial related presentations / publications
Public notes

Contacts
Principal investigator
Name 0 0
Address 0 0
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for public queries
Name 0 0
Sponsor Contact
Address 0 0
Country 0 0
Phone 0 0
(858) 732-3880
Fax 0 0
Email 0 0
Contact person for scientific queries

Data sharing statement
Will individual participant data (IPD) for this trial be available (including data dictionaries)?
Undecided
No/undecided IPD sharing reason/comment


What supporting documents are/will be available?

No Supporting Document Provided


Results publications and other study-related documents

No documents have been uploaded by study researchers.